

HY-15816 · Free Sample (0.1 - 0.2 mg)
MedChemExpress · Cat: HY-15816
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Manufacturer product page
medchemexpress.com/VRT752271.html
Description
Ulixertinib BVD-523; VRT752271 is a potent, orally active, highly selective, ATP-competitive and reversible covalent inhibitor of ERK1/2 kinases, with an IC50 of 0.3 nM against ERK2. Ulixertinib BVD-523; VRT752271 inhibits the phosphorylated ERK2 pERK and downstream kinase RSK pRSK in an A375 melanoma cell line.







