GENERAL CATALOGUE
GXH-II-052
HY-150684 · 50 mg
MedChemExpress · Cat: HY-150684
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medchemexpress.com/gxh-ii-052.htmlCatalog No: HY-150684
CAS No: 3031654-49-3
Category: Epigenetics
Pack Size: 50 mg
Brand: MedChemExpress
Description
GXH-II-052 is a potent bivalent bromodomain and extraterminal domain BET inhibitor. GXH-II-052 shows binding potential for BRD4-1, BRD4-2, BRD4-T, BRDT-1, BRDT-2, BRDT-T with Kd values of 28, 9.1, 4.8, 0.6, 8.4, 2.6 nM, respectively. GXH-II-052 shows antiproliferative activity. GXH-II-052 decreases the expression of c-Myc.