

HY-47573 · 10 mM * 1 mL in DMSO
MedChemExpress · Cat: HY-47573
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Manufacturer product page
medchemexpress.com/ccg273441.html
Description
CCG273441 is a covalent inhibitor of G protein-coupled receptor GPCR kinase 5 GRK5 with an IC50 value of 3.8 nM. CCG273441 is highly selective to GRK5 over GRK2 IC50=4.8 ?M by binding Cys474, a GRK5 subfamily-specific residue, as a covalent handle.







