

ab120282 · 10 mg
Verified Partner
Sign in to see pricing and request a quote.
Brand Store Product
No external links. Get your quote directly here.

Description
MW 357.8 Da, Purity >98 %. Selective blocker of NaV1.8 channels IC50 = 8 nM for human NaV1.8 . Shows greater than 100-fold selectivity over human NaV1.2, NaV1.3, NaV1.5, and NaV1.7 IC50 values =1 muM . Shows no significant activity against TRPV1, P2X2/3, CaV2.2 and KCNQ2/3 channels. Antinociceptive.