

ab146023 · 10 mg
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Description
MW 462.5 Da, Purity >98 %. Potent, selective, cell-permeable STAT3 inhibitor Kd = 880 nM . Inhibits STAT3 dimerization IC50 values are 0.28 and 10 muM for STAT3 SH2 domain-mediated ligand binding and STAT1 ligand binding, respectively . Blocks TRAIL-induced invasion.






